| 
|---|
 | mAChRsTooltip Muscarinic acetylcholine receptors | | Agonists |  | 
|---|
 | Antagonists |  - 3-Quinuclidinyl benzilate
  - 4-DAMP
  - Aclidinium bromide (+formoterol)
  - Abediterol
  - AF-DX 250
  - AF-DX 384
  - Ambutonium bromide
  - Anisodamine
  - Anisodine
  - Antihistamines (first-generation) (e.g., brompheniramine, buclizine, captodiame, chlorphenamine (chlorpheniramine), cinnarizine, clemastine, cyproheptadine, dimenhydrinate, dimetindene, diphenhydramine, doxylamine, meclizine, mequitazine, perlapine, phenindamine, pheniramine, phenyltoloxamine, promethazine, propiomazine, triprolidine)
  - AQ-RA 741
  - Atropine
  - Atropine methonitrate
  - Atypical antipsychotics (e.g., clozapine, fluperlapine, olanzapine (+fluoxetine), rilapine, quetiapine, tenilapine, zotepine)
  - Benactyzine
  - Benzatropine (benztropine)
  - Benzilone
  - Benzilylcholine mustard
  - Benzydamine
  - Bevonium
  - BIBN 99
  - Biperiden
  - Bornaprine
  - Camylofin
  - CAR-226,086
  - CAR-301,060
  - CAR-302,196
  - CAR-302,282
  - CAR-302,368
  - CAR-302,537
  - CAR-302,668
  - Caramiphen
  - Cimetropium bromide
  - Clidinium bromide
  - Cloperastine
  - CS-27349
  - Cyclobenzaprine
  - Cyclopentolate
  - Darifenacin
  - DAU-5884
  - Desfesoterodine
  - Dexetimide
  - DIBD
  - Dicycloverine (dicyclomine)
  - Dihexyverine
  - Difemerine
  - Diphemanil metilsulfate
  - Ditran
  - Drofenine
  - EA-3167
  - EA-3443
  - EA-3580
  - EA-3834
  - Emepronium bromide
  - Etanautine
  - Etybenzatropine (ethybenztropine)
  - Fenpiverinium
  - Fentonium bromide
  - Fesoterodine
  - Flavoxate
  - Glycopyrronium bromide (+beclometasone/formoterol, +indacaterol, +neostigmine)
  - Hexahydrodifenidol
  - Hexahydrosiladifenidol
  - Hexbutinol
  - Hexocyclium
  - Himbacine
  - HL-031,120
  - Homatropine
  - Imidafenacin
  - Ipratropium bromide (+salbutamol)
  - Isopropamide
  - J-104,129
  - Hyoscyamine
  - Mamba toxin 3
  - Mamba toxin 7
  - Mazaticol
  - Mebeverine
  - Meladrazine
  - Mepenzolate
  - Methantheline
  - Methoctramine
  - Methylatropine
  - Methylhomatropine
  - Methylscopolamine
  - Metixene
  - Muscarinic toxin 7
  - N-Ethyl-3-piperidyl benzilate
  - N-Methyl-3-piperidyl benzilate
  - Nefopam
  - Octatropine methylbromide (anisotropine methylbromide)
  - Orphenadrine
  - Otenzepad (AF-DX 116)
  - Otilonium bromide
  - Oxapium iodide
  - Oxitropium bromide
  - Oxybutynin
  - Oxyphencyclimine
  - Oxyphenonium bromide
  - PBID
  - PD-102,807
  - PD-0298029
  - Penthienate
  - Pethidine
  - pFHHSiD
  - Phenglutarimide
  - Phenyltoloxamine
  - Pipenzolate bromide
  - Piperidolate
  - Pirenzepine
  - Piroheptine
  - Pizotifen
  - Poldine
  - Pridinol
  - Prifinium bromide
  - Procyclidine
  - Profenamine (ethopropazine)
  - Propantheline bromide
  - Propiverine
  - Quinidine
  - 3-Quinuclidinyl thiochromane-4-carboxylate
  - Revefenacin
  - Rociverine
  - RU-47,213
  - SCH-57,790
  - SCH-72,788
  - SCH-217,443
  - Scopolamine (hyoscine)
  - Scopolamine butylbromide (hyoscine butylbromide)
  - Silahexacyclium
  - Sofpironium bromide
  - Solifenacin
  - SSRIsTooltip Selective serotonin reuptake inhibitors (e.g., femoxetine, paroxetine)
  - Telenzepine
  - Terodiline
  - Tetracyclic antidepressants (e.g., amoxapine, maprotiline, mianserin, mirtazapine)
  - Tiemonium iodide
  - Timepidium bromide
  - Tiotropium bromide
  - Tiquizium bromide
  - Tofenacin
  - Tolterodine
  - Tricyclic antidepressants (e.g., amitriptyline (+perphenazine), amitriptylinoxide, butriptyline, cidoxepin, clomipramine, desipramine, desmethyldesipramine, dibenzepin, dosulepin (dothiepin), doxepin, imipramine, lofepramine, nitroxazepine, northiaden (desmethyldosulepin), nortriptyline, protriptyline, quinupramine, trimipramine)
  - Tridihexethyl
  - Trihexyphenidyl
  - Trimebutine
  - Tripitamine (tripitramine)
  - Tropacine
  - Tropatepine
  - Tropicamide
  - Tropine benzilate
  - Trospium chloride
  - Typical antipsychotics (e.g., chlorpromazine, chlorprothixene, cyamemazine (cyamepromazine), loxapine, mesoridazine, thioridazine)
  - Umeclidinium bromide (+vilanterol)
  - WIN-2299
  - Xanomeline
  - Zamifenacin
     | 
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  | 
|---|
 Precursors (and prodrugs) |  | 
|---|
  - See also
  - Receptor/signaling modulators
  - Nicotinic acetylcholine receptor modulators
  - Acetylcholine metabolism/transport modulators
     |  
    | 
|---|
 | nAChRsTooltip Nicotinic acetylcholine receptors | Agonists (and PAMsTooltip positive allosteric modulators) |  - 5-HIAA
  - 6-Chloronicotine
  - A-84,543
  - A-366,833
  - A-582,941
  - A-867,744
  - ABT-202
  - ABT-418
  - ABT-560
  - ABT-894
  - Acetylcholine
  - Altinicline
  - Anabasine
  - Anatabine
  - Anatoxin-a
  - AR-R17779
  - Bephenium hydroxynaphthoate
  - Butinoline
  - Butyrylcholine
  - Carbachol
  - Choline
  - Choline m-bromophenyl ether
  - Cotinine
  - Cytisine
  - Decamethonium
  - Desformylflustrabromine
  - Dianicline
  - Dimethylphenylpiperazinium
  - Epibatidine
  - Epiboxidine
  - Ethanol (alcohol)
  - Ethoxysebacylcholine
  - EVP-4473
  - EVP-6124
  - Galantamine
  - GTS-21
  - Ispronicline
  - Ivermectin
  - JNJ-39393406
  - Levamisole
  - Lobeline
  - MEM-63,908 (RG-3487)
  - Morantel
  - Nicotine (tobacco)
  - NS-1738
  - PHA-543,613
  - PHA-709,829
  - PNU-120,596
  - PNU-282,987
  - Pozanicline
  - Pyrantel
  - Rivanicline
  - RJR-2429
  - Sazetidine A
  - SB-206553
  - Sebacylcholine
  - SIB-1508Y
  - SIB-1553A
  - SSR-180,711
  - Suberyldicholine
  - Suxamethonium (succinylcholine)
  - Suxethonium (succinyldicholine)
  - TC-1698
  - TC-1734
  - TC-1827
  - TC-2216
  - TC-5214
  - TC-5619
  - TC-6683
  - Tebanicline
  - Tribendimidine
  - Tropisetron
  - UB-165
  - Varenicline
  - WAY-317,538
  - XY-4083
     | 
|---|
 Antagonists (and NAMsTooltip negative allosteric modulators) |  | 
|---|
 
  | 
|---|
 Precursors (and prodrugs) |  | 
|---|
  - See also
  - Receptor/signaling modulators
  - Muscarinic acetylcholine receptor modulators
  - Acetylcholine metabolism/transport modulators
     |  
     |